Quantity: 50 MG
10 in stock
Product name: [Chx2]EM
Modifications: 1-aminocyclohexane-1-carboxlylic acid (Chx),
Purity: 95% by HPLC
Counter ion: Trifluoacetate
Format: Lyophilized powder
Description: [Chx2]EM2, an EM2 analogue substituting 1-aminocyclohexane-1-carboxlylic acid (Chx) for Pro. X-ray diffraction analysis revealed that [Chx2]EM2 is folded into the trans-form of Tyr–Chx. The manner of folding resembled that seen in D-TIPP, an EM analogue incorporating tetrahydroisoquinoline carboxylic acid, as well as the β-turn of Leu-enkephalin. Selectivity for the opioid μ-receptor was fairly well conserved by [Chx2]EM, suggesting that the folded form is important for μ-selectivity.
Usage: For Scientific Research Use Only, Not for Human Use.